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Drug
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No.
Drug (Description in trials)
DrugBank
KEGG DRUG
KEGG GENES
KEGG PATHWAY
Disease ID
1
Bosentan
[1]
Bosentan
Bosentan
[2]
Bosentan
Bosentan
,
Bosentan
💬
1.
Bosentan
×
Name
Other Names
Bosentan
Bosentan (USAN)
Bosentan hydrate (JAN)
Tracleer (TN)
Bosentan
Bosentan (INN)
[2]
EDNRA
EDNRA
,
EDNRB
💬
1.
Bosentan
×
Name
Full Name
EDNRA
endothelin receptor type A
EDNRB
endothelin receptor type B
[9]
Calcium signaling pathway
Calcium signaling pathway
,
Melanogenesis
,
Neuroactive ligand-receptor interaction
,
Pathways in cancer
,
Relaxin signaling pathway
,
Renin secretion
,
Vascular smooth muscle contraction
,
cAMP signaling pathway
,
cGMP-PKG signaling pathway
💬
[9]
Calcium signaling pathway
,
Melanogenesis
,
Neuroactive ligand-receptor interaction
,
Pathways in c
...
[10]
41
41
,
47
,
51
,
84
,
85
,
86
,
88
,
210
,
211
,
212
💬
1.
Bosentan
×
Disease ID
Name
41
Giant cell arteritis
47
Buerger disease
51
Scleroderma
84
Sarcoidosis
85
Idiopathic interstitial pneumonia
86
Pulmonary arterial hypertension
88
Chronic thromboembolic pulmonary hypertension
210
Single Ventricle
211
Hypoplastic left heart syndrome
212
Tricuspid atresia
2
Bosentan
(Tracleer)
[1]
Bosentan
Bosentan
[2]
Bosentan
Bosentan
,
Bosentan
💬
2.
Bosentan
(Tracleer)
×
Name
Other Names
Bosentan
Bosentan (USAN)
Bosentan hydrate (JAN)
Tracleer (TN)
Bosentan
Bosentan (INN)
[2]
EDNRA
EDNRA
,
EDNRB
💬
2.
Bosentan
(Tracleer)
×
Name
Full Name
EDNRA
endothelin receptor type A
EDNRB
endothelin receptor type B
[9]
Calcium signaling pathway
Calcium signaling pathway
,
Melanogenesis
,
Neuroactive ligand-receptor interaction
,
Pathways in cancer
,
Relaxin signaling pathway
,
Renin secretion
,
Vascular smooth muscle contraction
,
cAMP signaling pathway
,
cGMP-PKG signaling pathway
💬
[9]
Calcium signaling pathway
,
Melanogenesis
,
Neuroactive ligand-receptor interaction
,
Pathways in c
...
[1]
51
51
💬
2.
Bosentan
(Tracleer)
×
Disease ID
Name
51
Scleroderma
3
Bosentan
125 mg
[1]
Bosentan
Bosentan
[2]
Bosentan
Bosentan
,
Bosentan
💬
3.
Bosentan
125 mg
×
Name
Other Names
Bosentan
Bosentan (USAN)
Bosentan hydrate (JAN)
Tracleer (TN)
Bosentan
Bosentan (INN)
[2]
EDNRA
EDNRA
,
EDNRB
💬
3.
Bosentan
125 mg
×
Name
Full Name
EDNRA
endothelin receptor type A
EDNRB
endothelin receptor type B
[9]
Calcium signaling pathway
Calcium signaling pathway
,
Melanogenesis
,
Neuroactive ligand-receptor interaction
,
Pathways in cancer
,
Relaxin signaling pathway
,
Renin secretion
,
Vascular smooth muscle contraction
,
cAMP signaling pathway
,
cGMP-PKG signaling pathway
💬
[9]
Calcium signaling pathway
,
Melanogenesis
,
Neuroactive ligand-receptor interaction
,
Pathways in c
...
[1]
51
51
💬
3.
Bosentan
125 mg
×
Disease ID
Name
51
Scleroderma
4
Bosentan
62.5 mg
[1]
Bosentan
Bosentan
[2]
Bosentan
Bosentan
,
Bosentan
💬
4.
Bosentan
62.5 mg
×
Name
Other Names
Bosentan
Bosentan (USAN)
Bosentan hydrate (JAN)
Tracleer (TN)
Bosentan
Bosentan (INN)
[2]
EDNRA
EDNRA
,
EDNRB
💬
4.
Bosentan
62.5 mg
×
Name
Full Name
EDNRA
endothelin receptor type A
EDNRB
endothelin receptor type B
[9]
Calcium signaling pathway
Calcium signaling pathway
,
Melanogenesis
,
Neuroactive ligand-receptor interaction
,
Pathways in cancer
,
Relaxin signaling pathway
,
Renin secretion
,
Vascular smooth muscle contraction
,
cAMP signaling pathway
,
cGMP-PKG signaling pathway
💬
[9]
Calcium signaling pathway
,
Melanogenesis
,
Neuroactive ligand-receptor interaction
,
Pathways in c
...
[1]
51
51
💬
4.
Bosentan
62.5 mg
×
Disease ID
Name
51
Scleroderma
5
Bosentan
administration
[1]
Bosentan
Bosentan
[2]
Bosentan
Bosentan
,
Bosentan
💬
5.
Bosentan
administration
×
Name
Other Names
Bosentan
Bosentan (USAN)
Bosentan hydrate (JAN)
Tracleer (TN)
Bosentan
Bosentan (INN)
[2]
EDNRA
EDNRA
,
EDNRB
💬
5.
Bosentan
administration
×
Name
Full Name
EDNRA
endothelin receptor type A
EDNRB
endothelin receptor type B
[9]
Calcium signaling pathway
Calcium signaling pathway
,
Melanogenesis
,
Neuroactive ligand-receptor interaction
,
Pathways in cancer
,
Relaxin signaling pathway
,
Renin secretion
,
Vascular smooth muscle contraction
,
cAMP signaling pathway
,
cGMP-PKG signaling pathway
💬
[9]
Calcium signaling pathway
,
Melanogenesis
,
Neuroactive ligand-receptor interaction
,
Pathways in c
...
[1]
86
86
💬
5.
Bosentan
administration
×
Disease ID
Name
86
Pulmonary arterial hypertension
6
Bosentan
and Sildenafil
[2]
Bosentan
Bosentan
,
Sildenafil
[3]
Bosentan
Bosentan
,
Bosentan
,
Sildenafil
💬
6.
Bosentan
and Sildenafil
×
Name
Other Names
Bosentan
Bosentan (USAN)
Bosentan hydrate (JAN)
Tracleer (TN)
Bosentan
Bosentan (INN)
Sildenafil
Sildenafil (INN)
Aphrodil (TN)
[3]
EDNRA
EDNRA
,
EDNRB
,
PDE5A
💬
6.
Bosentan
and Sildenafil
×
Name
Full Name
EDNRA
endothelin receptor type A
EDNRB
endothelin receptor type B
PDE5A
phosphodiesterase 5A
[11]
Calcium signaling pathway
Calcium signaling pathway
,
Melanogenesis
,
Metabolic pathways
,
Neuroactive ligand-receptor interaction
,
Pathways in cancer
,
Purine metabolism
,
Relaxin signaling pathway
,
Renin secretion
,
Vascular smooth muscle contraction
,
cAMP signaling pathway
,
cGMP-PKG signaling pathway
💬
[11]
Calcium signaling pathway
,
Melanogenesis
,
Metabolic pathways
,
Neuroactive ligand-receptor inter
...
[1]
86
86
💬
6.
Bosentan
and Sildenafil
×
Disease ID
Name
86
Pulmonary arterial hypertension
7
Bosentan
group
[1]
Bosentan
Bosentan
[2]
Bosentan
Bosentan
,
Bosentan
💬
7.
Bosentan
group
×
Name
Other Names
Bosentan
Bosentan (USAN)
Bosentan hydrate (JAN)
Tracleer (TN)
Bosentan
Bosentan (INN)
[2]
EDNRA
EDNRA
,
EDNRB
💬
7.
Bosentan
group
×
Name
Full Name
EDNRA
endothelin receptor type A
EDNRB
endothelin receptor type B
[9]
Calcium signaling pathway
Calcium signaling pathway
,
Melanogenesis
,
Neuroactive ligand-receptor interaction
,
Pathways in cancer
,
Relaxin signaling pathway
,
Renin secretion
,
Vascular smooth muscle contraction
,
cAMP signaling pathway
,
cGMP-PKG signaling pathway
💬
[9]
Calcium signaling pathway
,
Melanogenesis
,
Neuroactive ligand-receptor interaction
,
Pathways in c
...
[1]
51
51
💬
7.
Bosentan
group
×
Disease ID
Name
51
Scleroderma
8
BOSENTAN
MONOHIDRATO
[1]
Bosentan
Bosentan
[2]
Bosentan
Bosentan
,
Bosentan
💬
8.
BOSENTAN
MONOHIDRATO
×
Name
Other Names
Bosentan
Bosentan (USAN)
Bosentan hydrate (JAN)
Tracleer (TN)
Bosentan
Bosentan (INN)
[2]
EDNRA
EDNRA
,
EDNRB
💬
8.
BOSENTAN
MONOHIDRATO
×
Name
Full Name
EDNRA
endothelin receptor type A
EDNRB
endothelin receptor type B
[9]
Calcium signaling pathway
Calcium signaling pathway
,
Melanogenesis
,
Neuroactive ligand-receptor interaction
,
Pathways in cancer
,
Relaxin signaling pathway
,
Renin secretion
,
Vascular smooth muscle contraction
,
cAMP signaling pathway
,
cGMP-PKG signaling pathway
💬
[9]
Calcium signaling pathway
,
Melanogenesis
,
Neuroactive ligand-receptor interaction
,
Pathways in c
...
[1]
86
86
💬
8.
BOSENTAN
MONOHIDRATO
×
Disease ID
Name
86
Pulmonary arterial hypertension
9
Bosentan
monohydrat
[1]
Bosentan
Bosentan
[2]
Bosentan
Bosentan
,
Bosentan
💬
9.
Bosentan
monohydrat
×
Name
Other Names
Bosentan
Bosentan (USAN)
Bosentan hydrate (JAN)
Tracleer (TN)
Bosentan
Bosentan (INN)
[2]
EDNRA
EDNRA
,
EDNRB
💬
9.
Bosentan
monohydrat
×
Name
Full Name
EDNRA
endothelin receptor type A
EDNRB
endothelin receptor type B
[9]
Calcium signaling pathway
Calcium signaling pathway
,
Melanogenesis
,
Neuroactive ligand-receptor interaction
,
Pathways in cancer
,
Relaxin signaling pathway
,
Renin secretion
,
Vascular smooth muscle contraction
,
cAMP signaling pathway
,
cGMP-PKG signaling pathway
💬
[9]
Calcium signaling pathway
,
Melanogenesis
,
Neuroactive ligand-receptor interaction
,
Pathways in c
...
[1]
86
86
💬
9.
Bosentan
monohydrat
×
Disease ID
Name
86
Pulmonary arterial hypertension
10
BOSENTAN
MONOHYDRATE
[1]
Bosentan
Bosentan
[2]
Bosentan
Bosentan
,
Bosentan
💬
10.
BOSENTAN
MONOHYDRATE
×
Name
Other Names
Bosentan
Bosentan (USAN)
Bosentan hydrate (JAN)
Tracleer (TN)
Bosentan
Bosentan (INN)
[2]
EDNRA
EDNRA
,
EDNRB
💬
10.
BOSENTAN
MONOHYDRATE
×
Name
Full Name
EDNRA
endothelin receptor type A
EDNRB
endothelin receptor type B
[9]
Calcium signaling pathway
Calcium signaling pathway
,
Melanogenesis
,
Neuroactive ligand-receptor interaction
,
Pathways in cancer
,
Relaxin signaling pathway
,
Renin secretion
,
Vascular smooth muscle contraction
,
cAMP signaling pathway
,
cGMP-PKG signaling pathway
💬
[9]
Calcium signaling pathway
,
Melanogenesis
,
Neuroactive ligand-receptor interaction
,
Pathways in c
...
[4]
51
51
,
84
,
86
,
88
💬
10.
BOSENTAN
MONOHYDRATE
×
Disease ID
Name
51
Scleroderma
84
Sarcoidosis
86
Pulmonary arterial hypertension
88
Chronic thromboembolic pulmonary hypertension